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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T14194 | β-NETA | α-NETA | AChE |
β-NETA (α-NETA) is a stable, noncompetitive, slowly reversible choline acetyltransferase (ChAT) inhibitor with an IC50 of 9 μM and is a potent chemokine-like receptor-1 (CMKLR1) antagonist. β-NETA has anti-cancer activit... | |||
T3767 | Polygalacic acid | Virgaureagenin G | MMP , AChR , AChE |
Polygalacic acid (Virgaureagenin G)(PA) significantly improves cholinergic system reactivity, as indicated by decreased acetylcholinesterase (AChE) activity, increases choline acetyltransferase (ChAT) activity, and eleva... | |||
T29963 | Americanol A | ||
Americanol A enhances choline acetyltransferase activity; has neurotrophic properties. | |||
T13975 | ZSET-845 | Others | |
ZSET-845 is an enhancer of cognitive which enhances choline acetyltransferase activity in the hippocampus in the rat. | |||
T29203 | Zanapezil fumarate | TAK 147,TAK147,TAK-147 | |
Zanapezil is an acetylcholinesterase (AChE) inhibitor. Zanapezil increases choline acetyltransferase activity in cultured rat septal cholinergic neurons. | |||
T4497L | Amifampridine phosphate | BRN0110232,3,6-DAP,SC10,BRN 0110232,BRN-0110232,NSC 521760 | |
Amifampridine is mainly used to treat many rare muscle diseases. In the United States, aminopyridine is being studied for the treatment of Lambert-Eaton myasmus syndrome (LEMS). Amifampridine is also used to treat many c... | |||
T61454 | α-NETA | ||
α-NETA is a potent and noncompetitive choline acetyltransferase (ChA) inhibitor with an IC 50 of 9 μM. α-NETA is a potent ALDH1A1 ( IC 50 =0.04 μM) and chemokine-like receptor-1 (CMKLR1) antagonist. α-NETA weakly inhibit... |